-Конъюгаты антибиотиков с антителами: рациональный дизайн для улучшения фармакологических свойств

January 6, 2020 — December 31, 2022

Korshun V.A. (PI)

Laboratory of molecular design and synthesis

Grant, RFBR

List of publications

  1. Sapozhnikova KA, Misyurin AV, Pestov NB, Meleshkina EG, Oreshkov SD, Ganzhula EP, Mikhailova AS, Korshun VA, Misyurin VA, Brylev VA (2021). Detection of the PRAME Protein on the Surface of Melanoma Cells Using a Fluorescently Labeled Monoclonal Antibody. Russ. J. Bioorganic Chem. 47 (5), 1077–1085
  2. Sapozhnikova KA, Misyurin VA, Ryazantsev DY, Kokin EA, Finashutina YP, Alexeeva AV, Ivanov IA, Kocharovskaya MV, Tikhonova NA, Popova GP, Alferova VA, Ustinov AV, Korshun VA, Brylev VA (2021). Sensitive Immunofluorescent Detection of the PRAME Antigen Using a Practical Antibody Conjugation Approach. Int J Mol Sci 22 (23), 12845
  3. Sapozhnikova KA, Gulyak EL, Misyurin VA, Simonova MA, Ryabukhina EV, Alexeeva AV, Tikhonova NA, Lyzhko NA, Popova GP, Misyurin AV, Ustinov AV, Korshun VA, Alferova VA, Ryazantsev DY, Brylev VA (2023). Branched Linkers for Site-Specific Fluorescent Labeling of Antibodies. Molecules 28 (1), 425
  4. Sapozhnikova KA, Gulyak EL, Brylev VA, Misyurin VA, Oreshkov SD, Alexeeva AV, Ryazantsev DY, Simonova MA, Ryabukhina EV, Popova GP, Tikhonova NA, Lyzhko NA, Barmashov AE, Misyurin AV, Ustinov AV, Alferova VA, Korshun VA (2023). Aminooxy Click Modification of a Periodate-Oxidized Immunoglobulin G: A General Approach to Antibody–Drug Conjugates with Dye-Mediated Expeditious Stoichiometry Control. Int J Mol Sci 24 (6), 5134
  5. Alferova VA, Maviza TP, Biryukov MV, Zakalyukina YV, Lukianov DA, Skvortsov DA, Vasilyeva LA, Tashlitsky VN, Polshakov VI, Sergiev PV, Korshun VA, Osterman IA (2022). Biological evaluation and spectral characterization of a novel tetracenomycin X congener. Biochimie 192, 63–71
  6. Veryutin DA, Doroshenko IA, Martynova EA, Sapozhnikova KA, Svirshchevskaya EV, Shibaeva AV, Markova AA, Chistov AA, Borisova NE, Shuvalov MV, Korshun VA, Alferova VA, Podrugina TA (2023). Probing tricarbocyanine dyes for targeted delivery of anthracyclines. Biochimie 206, 12–23